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PD153035 hydrochloride
CAS No. 183322-45-4
PD153035 hydrochloride ( AG-1517 )
Catalog No. M12831 CAS No. 183322-45-4
PD153035 hydrochloride (ZM 252868; AG 1517) is a potent and specific inhibitor of EGFR with Ki and IC50 of 5.2 pM and 29 pM; little effect against PGDFR, FGFR, CSF-1, InsR and Src.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 42 | In Stock |
|
| 10MG | 56 | In Stock |
|
| 25MG | 113 | In Stock |
|
| 50MG | 221 | In Stock |
|
| 100MG | 375 | In Stock |
|
| 500MG | 853 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePD153035 hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionPD153035 hydrochloride (ZM 252868; AG 1517) is a potent and specific inhibitor of EGFR with Ki and IC50 of 5.2 pM and 29 pM; little effect against PGDFR, FGFR, CSF-1, InsR and Src.
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DescriptionPD153035 hydrochloride (ZM 252868; AG 1517) is a potent and specific inhibitor of EGFR with Ki and IC50 of 5.2 pM and 29 pM; little effect against PGDFR, FGFR, CSF-1, InsR and Src.
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SynonymsAG-1517
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PathwayAngiogenesis
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TargetEGFR
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RecptorEGFR; EGFR
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number183322-45-4
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Formula Weight396.67
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Molecular FormulaC16H15BrClN3O2
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Purity>98%(HPLC)
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SolubilityDMSO: 0.5 mg/mL (1.26 mM)
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SMILESCOc(c1)c(OC)cc2c1ncnc2Nc3cc(Br)ccc3.Cl
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Chemical NameN-(3-bromophenyl)-6,7-dimethoxyquinazolin-4-amine hydrochloride
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Fry DW, et al. Science. 1994, 265(5175), 1093-1095.
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